Telmisartan-d4
Referencia HY-13955S1-1mg
embalaje : 1mg
Marca : MedChemExpress
Telmisartan-d4 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM[1][2].
Para uso exclusivo en investigación. No vendemos a pacientes.
Telmisartan-d4 Estructura química
This product is a controlled substance and not for sale in your territory.
Ver todos los productos específicos de isoformas Angiotensin Receptor:
Descripciòn |
Telmisartan-d4 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM[1][2]. |
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In Vitro |
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1]. MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. |
Peso molecular |
518.64 |
Fòrmula |
C33H26D4N4O2 |
Unlabeled CAS |
144701-48-4 |
SMILES |
CCCC1=NC2=C(C)C=C(C3=NC4=CC=CC=C4N3C)C=C2N1CC5=C([2H])C([2H])=C(C6=CC=CC=C6C(O)=O)C([2H])=C5[2H] |
Envío | Room temperature in continental US; may vary elsewhere. |
Almacenamiento |
Please store the product under the recommended conditions in the Certificate of Analysis. |
Pureza y Documentación | |
Referencias |
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Telmisartan-d4 Related Classifications
- Endocrinology Cardiovascular Disease
- Others GPCR/G Protein Autophagy
- Isotope-Labeled Compounds Angiotensin Receptor Autophagy
Calculadora de molaridad
Calculadora de dilución
The molarity calculator equation
Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)
The dilution calculator equation
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2
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Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.
Keywords:
Telmisartan-d4Isotope-Labeled CompoundsAngiotensin ReceptorAutophagyInhibitorinhibitorinhibit