AR-C155858 [496791-37-8]
Referência HY-13248-1mg
Tamanho : 1mg
Marca : MedChemExpress
AR-C155858 is a selective monocarboxylate transporter MCT1 and MCT2 inhibitor with Kis of 2.3 nM and 10 nM, respectively.
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AR-C155858 Chemical Structure
CAS No. : 496791-37-8
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Based on 38 publication(s) in Google Scholar
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AR-C155858 purchased from MedChemExpress. Usage Cited in: Am J Physiol Cell Physiol. 2016 Jul 1;311(1):C116-26. [Abstract]
- Inhibition of pyruvate transport in HEK293 cells. Summary of 24 cells in three separate experiments.
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AR-C155858 purchased from MedChemExpress. Usage Cited in: Oncotarget. 2014 Nov 30;5(22):11029-37. [Abstract]
- The MCT1/2 inhibitor AR-C155858 significantly reduces mammosphere formation in MDA-MB-231 cells. Note that AR-C155858 also effectively reduces mammosphere formation in this cellular context, with an IC50 of ~1-2 μM. The vehicle-alone control is normalized to one.